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Number of items: 32.

Stubba, Daniel ; Bensinger, Dennis ; Steinbacher, Janika ; Proskurjakov, Lilia ; Salcedo Gómez, Álvaro ; Schmidt, Uwe ; Roth, Stefan ; Schmitz, Katja ; Schmidt, Boris (2019):
Cell‐Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit.
In: ChemMedChem, 14 (23), pp. 2005-2022. ISSN 1860-7179,
DOI: 10.1002/cmdc.201900472,
[Article]

Bensinger, Dennis ; Stubba, Daniel ; Cremer, Anjali ; Kohl, Vanessa ; Waßmer, Theresa ; Stuckert, Johanna ; Engemann, Victoria ; Stegmaier, Kimberly ; Schmitz, Katja ; Schmidt, Boris (2019):
Virtual Screening Identifies Irreversible FMS-like Tyrosine Kinase 3 Inhibitors with Activity toward Resistance-Conferring Mutations.
In: Journal of Medicinal Chemistry, 62 (5), pp. 2428-2446. American Chemical Society, ISSN 0022-2623,
DOI: 10.25534/tuprints-00009651,
[Article]

Bensinger, Dennis ; Neumann, Theresa ; Scholz, Christoph ; Voss, Constantin ; Knorr, Sabine ; Kuckelkorn, Ulrike ; Hamacher, Kay ; Kloetzel, Peter-Michael ; Schmidt, Boris (2016):
Elastase-like Activity Is Dominant to Chymotrypsin-like Activity in 20S Proteasome's β5 Catalytic Subunit.
In: ACS chemical biology, 11 (7), pp. 1800-1804. ISSN 1554-8937,
[Article]

Scholz, Christoph ; Knorr, Sabine ; Hamacher, Kay ; Schmidt, Boris (2015):
DOCKTITE-A Highly Versatile Step-by-Step Workflow for Covalent Docking and Virtual Screening in the Molecular Operating Environment.
In: Journal of chemical information and modeling, 55 (2), pp. 398-406. ISSN 1549-960X,
[Article]

Neumann, Theresa ; Benajiba, Lina ; Göring, Stefan ; Stegmaier, Kimberly ; Schmidt, Boris (2015):
Evaluation of Improved Glycogen Synthase Kinase-3α Inhibitors in Models of Acute Myeloid Leukemia.
In: Journal of Medicinal Chemistry, 58 (22), pp. 8907-8919. American Chemical Society, ISSN 0022-2623,
DOI: 10.25534/tuprints-00009652,
[Article]

Voss, Constantin ; Scholz, Christoph ; Knorr, Sabine ; Beck, Philipp ; Stein, Martin L. ; Zall, Andrea ; Kuckelkorn, Ulrike ; Kloetzel, Peter-Michael ; Groll, Michael ; Hamacher, Kay ; Schmidt, Boris (2014):
α-Keto Phenylamides as P1'-Extended Proteasome Inhibitors.
In: ChemMedChem, 9 (11), pp. 2557-2564. ISSN 1860-7187,
[Article]

Schupp, M. ; Lee, C. L. D. ; Frost, N. ; Umbreen, Sumaira ; Schmidt, Boris ; Unger, T. ; Kintscher, U. (2006):
CHBPR-Regulation of PPARg Activity by Losartan Metabolites.
In: Hypertension, 47, pp. 586-589. [Article]

Silva, Luiz Everson da ; Joussef, Antonio Carlos ; Foro, Sabine ; Schmidt, Boris (2005):
4-Fluoro-N-(quinolin-8-yl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (12), pp. o4387-o4388. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805039188,
[Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
4-Nitro-N-(8-quinolyl)-benzenesulfon-amide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11), pp. o3778-o3779. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805032691,
[Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
5 2,4,6-Triisopropyl-N-(8-quinolyl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11), pp. o3780-o3781. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805032708,
[Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
N-(5,7-Dibromo-8-quinolyl)-4-fluoro-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11), pp. o3782-o3783. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S160053680503271X,
[Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
5,7-Dibromo-N-tosyl-quinolin-8-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (10), pp. o3435-o3436. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S160053680502773X,
[Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
6-Nitroquinolin-2(1H)-one.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (9), pp. o2992-o2993. Wiley, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805025894,
[Article]

Braun, Hannes R. ; Meusinger, Reinhard ; Schmidt, Boris (2005):
2-iodethanols from aldehydes, diiodomethane and iso-propylmagnesium chloride.
46, In: Tetrahedron Letters, pp. 2551-2554. [Article]

Schmidt, Boris ; Narlawar, Rajeshwar ; Braun, Hannes (2005):
Drug Development and PET-Diagnostics for Alzheimer's Disease.
In: Current Medicinal Chemistry, 12, pp. 1677-1695. [Article]

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005):
N-Benzyl-8-nitroquinolin-2-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, 61, pp. o3837-o3838. [Article]

Braun, A. ; Umbreen, Sumaira ; Groll, M. ; Kuckelkorn, U. ; Mlynarczuk, I. ; Wiegand, M. E. ; Drung, I. ; Kloetzel, P. M. ; Schmidt, Boris (2005):
Tripeptide mimetics inhibit the 20S proteasome by covalent bonding to the active site threonines.
In: Journal of Biological Chemistry, 280, pp. 28394-28411. [Article]

Schmidt, Boris ; Siegler, Alexander (2004):
Aspartic Proteases involved in Alzheimer's disease.
In: Highlights in bioorganic chemistry. Eds.: Schmuck, Carsten ; Wennemers, Helma. - Weinheim : Wiley-VCH Verl. , 2004. S. 262-276 , ISBN 3-527-30656-0, Weinheim, Wiley-VCH Verl., [Book Section]

Schmidt, Boris ; Jiricek, Jan ; Titz, Alexander ; Ye, Guofeng ; Parang, Keykavous (2004):
Copper dipicolinates as peptidomimetic ligands for the Src SH2 domain.
In: Bioorganic & Medicinal Chemistry Letters, 14, pp. 4203-4206. [Article]

Schmidt, Boris ; Braun, Hannes A. (2004):
E-1,2-Dichlorovinyl ethers as irreversible protease inhibitors.
In: Tetrahydron Letterrs, 45, pp. 1751-1753. [Article]

Larbig, Gregor ; Zall, Andreas ; Schmidt, Boris (2004):
Inhibitors designed for presenilin 1 by means of aspartic acid activation : Preliminary Communication.
In: Helvetica Chimica Acta, 87, pp. 2334-2340. [Article]

Schmidt, Boris (2004):
[Rez.:] Molecular biology in medicinal chemistry / ed. by Th. Dingermann .... - Weinheim : Wiley-VCH, 2004 (Methods and principles in medicinal chemistry ; 21) ISBN 7-30431-2.
In: ChemBioChem, 5, pp. 1153-1154. [Article]

Schmidt, Boris ; Larbig, Gregor (2004):
[Rez.:] More targets, strategies, methods / K. C. Nicolaou and S. A. Snyder. - 2003. -(Classics in total synthesis / K. C. Nicolaou and S. A. Snyder ; 2) ISBN: 3-527-30685-4.
In: ChemBioChem (ISSN 1439-4227), 5, p. 885. [Article]

Schmidt, Boris ; Drexler, H. ; Schieffer, Bernhard (2004):
Therapeutic Effects of Angiotensin (AT1) Receptor Antagonists: Potential Contribution of Mechanisms Other Than AT1 Receptor Blockade.
In: American Journal of Cardiovascular Drugs, pp. 361-368. [Article]

Schmidt, Boris ; Drexler, Helmut ; Schieffer, Bernhard (2004):
Therapeutic effects of angiotensin (AT1) receptor antagonists : potential contribution of mechanisms other than AT1 receptor blockade.
4, In: American Journal of Cardiovascular Drugs, pp. 361-368. [Article]

Muller, Gilles ; Schmidt, Boris ; Jiricek, Jan ; Lbuenzli, Jean Claude G. ; Schenk, Kurt J. (2003):
3-[2,6-Bis(diethyl-carbamoyl)-pyridin-4-yl]-N-(tert-butoxycarbonyl)alanine methyl ester: a chiral tridentate ligand that causes a diastereomeric excess of its lanthanide complexes in solution.
In: Acta Crystallographica, Section C: Crystal Structure Communications, 59, pp. 353-356. [Article]

Schmidt, Boris ; Schieffer, Bernhard (2003):
Angiotensin II AT1 Receptor Antagonists : Clinical Implications of Active Metabolites.
In: Journal of Medicinal Chemistry, 46, p. 2261. [Article]

Schieffer, Bernhard ; Schmidt, Boris ; Drexler, H. (2003):
Angiotensin-II-Rezeptor-unabhängige anti-inflammatorische und antiaggregatorische Eigenschaften von AT1-Antagonisten. Rolle aktiver Metaboliten.
In: Herz BNK, 28, p. 2. [Article]

Schmidt, Boris (2003):
Aspartic Proteases involved in Alzheimer's disease.
In: ChemBioChem : a European journal of chemical biology, 4, pp. 367-378. [Article]

Schmidt, Boris (2003):
Selective inhibition of proteases :design of beta- and gamma-scretase inhibitors.
In: International conference on aspartic proteases and inhibitors <2003, Kyoto, Japan> : [proceedings], S. 20, [Conference or Workshop Item]

Schmidt, Boris ; Kühn, Christian ; Ehlert, Dennis K. ; Lindeberg, Gunnar ; Lindman, Susanne ; Karlén, Anders ; Hallberg, Anders (2003):
A frame shifted disulfide bridged analogue of angiotensin II.
In: Bioorganic medicinal chemistry, pp. 985-990. [Article]

Krämer, Christine ; Sunkomat, Julia ; Witte, Jane ; Luchtefeld, Maren ; Walden, Michael ; Schmidt, Boris ; Boger, Rainer H. ; Tsikas, Dimitrios ; Forssmann, Wolf-Georg ; Drexler, Helmut ; Schieffer, Bernhard (2002):
Angiotensin II receptor-independent antiinflammatory and antiaggregatory properties of Losartan : role of the active metabolite EXP3179.
In: Circulation Research, 90, pp. 770-777. [Article]

This list was generated on Tue Aug 3 04:48:45 2021 CEST.