2019

Bensinger, Dennis ; Stubba, Daniel ; Cremer, Anjali ; Kohl, Vanessa ; Waßmer, Theresa ; Stuckert, Johanna ; Engemann, Victoria ; Stegmaier, Kimberly ; Schmitz, Katja ; Schmidt, Boris (2019)
Virtual Screening Identifies Irreversible FMS-like Tyrosine Kinase 3 Inhibitors with Activity toward Resistance-Conferring Mutations.
In: Journal of Medicinal Chemistry, 62 (5)
doi: 10.1021/acs.jmedchem.8b01714
Artikel, Bibliographie

Stubba, Daniel ; Bensinger, Dennis ; Steinbacher, Janika ; Proskurjakov, Lilia ; Salcedo Gómez, Álvaro ; Schmidt, Uwe ; Roth, Stefan ; Schmitz, Katja ; Schmidt, Boris (2019)
Cell‐Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit.
In: ChemMedChem, 14 (23)
doi: 10.1002/cmdc.201900472
Artikel, Bibliographie

2016

Bensinger, Dennis ; Neumann, Theresa ; Scholz, Christoph ; Voss, Constantin ; Knorr, Sabine ; Kuckelkorn, Ulrike ; Hamacher, Kay ; Kloetzel, Peter-Michael ; Schmidt, Boris (2016)
Elastase-like Activity Is Dominant to Chymotrypsin-like Activity in 20S Proteasome's β5 Catalytic Subunit.
In: ACS chemical biology, 11 (7)
Artikel, Bibliographie

2015

Scholz, Christoph ; Knorr, Sabine ; Hamacher, Kay ; Schmidt, Boris (2015)
DOCKTITE-A Highly Versatile Step-by-Step Workflow for Covalent Docking and Virtual Screening in the Molecular Operating Environment.
In: Journal of chemical information and modeling, 55 (2)
Artikel, Bibliographie

Neumann, Theresa ; Benajiba, Lina ; Göring, Stefan ; Stegmaier, Kimberly ; Schmidt, Boris (2015)
Evaluation of Improved Glycogen Synthase Kinase-3α Inhibitors in Models of Acute Myeloid Leukemia.
In: Journal of Medicinal Chemistry, 58 (22)
Artikel, Bibliographie

2014

Voss, Constantin ; Scholz, Christoph ; Knorr, Sabine ; Beck, Philipp ; Stein, Martin L. ; Zall, Andrea ; Kuckelkorn, Ulrike ; Kloetzel, Peter-Michael ; Groll, Michael ; Hamacher, Kay ; Schmidt, Boris (2014)
α-Keto Phenylamides as P1'-Extended Proteasome Inhibitors.
In: ChemMedChem, 9 (11)
Artikel, Bibliographie

2006

Schupp, M. ; Lee, C. L. D. ; Frost, N. ; Umbreen, Sumaira ; Schmidt, Boris ; Unger, T. ; Kintscher, U. (2006)
CHBPR-Regulation of PPARg Activity by Losartan Metabolites.
In: Hypertension, 47
Artikel, Bibliographie

2005

Silva, Luiz Everson da ; Joussef, Antonio Carlos ; Foro, Sabine ; Schmidt, Boris (2005)
4-Fluoro-N-(quinolin-8-yl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (12)
doi: 10.1107/S1600536805039188
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
4-Nitro-N-(8-quinolyl)-benzenesulfon-amide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11)
doi: 10.1107/S1600536805032691
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
5 2,4,6-Triisopropyl-N-(8-quinolyl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11)
doi: 10.1107/S1600536805032708
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
N-(5,7-Dibromo-8-quinolyl)-4-fluoro-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (11)
doi: 10.1107/S160053680503271X
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
5,7-Dibromo-N-tosyl-quinolin-8-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (10)
doi: 10.1107/S160053680502773X
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
6-Nitroquinolin-2(1H)-one.
In: Acta Crystallographica, Section E: Structure Reports Online, 61 (9)
doi: 10.1107/S1600536805025894
Artikel, Bibliographie

Braun, Hannes R. ; Meusinger, Reinhard ; Schmidt, Boris (2005)
2-iodethanols from aldehydes, diiodomethane and iso-propylmagnesium chloride.
In: Tetrahedron Letters, 46
Artikel, Bibliographie

Schmidt, Boris ; Narlawar, Rajeshwar ; Braun, Hannes (2005)
Drug Development and PET-Diagnostics for Alzheimer's Disease.
In: Current Medicinal Chemistry, 12
Artikel, Bibliographie

Silva, Luiz Everson da ; Joussef, Antonio C. ; Foro, Sabine ; Schmidt, Boris (2005)
N-Benzyl-8-nitroquinolin-2-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, 61
Artikel, Bibliographie

Braun, A. ; Umbreen, Sumaira ; Groll, M. ; Kuckelkorn, U. ; Mlynarczuk, I. ; Wiegand, M. E. ; Drung, I. ; Kloetzel, P. M. ; Schmidt, Boris (2005)
Tripeptide mimetics inhibit the 20S proteasome by covalent bonding to the active site threonines.
In: Journal of Biological Chemistry, 280
Artikel, Bibliographie

2004

Schmidt, Boris ; Siegler, Alexander (2004)
Aspartic Proteases involved in Alzheimer's disease.
In: Highlights in bioorganic chemistry
Buchkapitel, Bibliographie

Schmidt, Boris ; Jiricek, Jan ; Titz, Alexander ; Ye, Guofeng ; Parang, Keykavous (2004)
Copper dipicolinates as peptidomimetic ligands for the Src SH2 domain.
In: Bioorganic & Medicinal Chemistry Letters, 14
Artikel, Bibliographie

Schmidt, Boris ; Braun, Hannes A. (2004)
E-1,2-Dichlorovinyl ethers as irreversible protease inhibitors.
In: Tetrahydron Letterrs, 45
Artikel, Bibliographie

Larbig, Gregor ; Zall, Andreas ; Schmidt, Boris (2004)
Inhibitors designed for presenilin 1 by means of aspartic acid activation : Preliminary Communication.
In: Helvetica Chimica Acta, 87
Artikel, Bibliographie

Schmidt, Boris (2004)
[Rez.:] Molecular biology in medicinal chemistry / ed. by Th. Dingermann .... - Weinheim : Wiley-VCH, 2004 (Methods and principles in medicinal chemistry ; 21) ISBN 7-30431-2.
In: ChemBioChem, 5
Artikel, Bibliographie

Schmidt, Boris ; Larbig, Gregor (2004)
[Rez.:] More targets, strategies, methods / K. C. Nicolaou and S. A. Snyder. - 2003. -(Classics in total synthesis / K. C. Nicolaou and S. A. Snyder ; 2) ISBN: 3-527-30685-4.
In: ChemBioChem (ISSN 1439-4227), 5
Artikel, Bibliographie

Schmidt, Boris ; Drexler, H. ; Schieffer, Bernhard (2004)
Therapeutic Effects of Angiotensin (AT1) Receptor Antagonists: Potential Contribution of Mechanisms Other Than AT1 Receptor Blockade.
In: American Journal of Cardiovascular Drugs
Artikel, Bibliographie

Schmidt, Boris ; Drexler, Helmut ; Schieffer, Bernhard (2004)
Therapeutic effects of angiotensin (AT1) receptor antagonists : potential contribution of mechanisms other than AT1 receptor blockade.
In: American Journal of Cardiovascular Drugs, 4
Artikel, Bibliographie

2003

Muller, Gilles ; Schmidt, Boris ; Jiricek, Jan ; Lbuenzli, Jean Claude G. ; Schenk, Kurt J. (2003)
3-[2,6-Bis(diethyl-carbamoyl)-pyridin-4-yl]-N-(tert-butoxycarbonyl)alanine methyl ester: a chiral tridentate ligand that causes a diastereomeric excess of its lanthanide complexes in solution.
In: Acta Crystallographica, Section C: Crystal Structure Communications, 59
Artikel, Bibliographie

Schmidt, Boris ; Schieffer, Bernhard (2003)
Angiotensin II AT1 Receptor Antagonists : Clinical Implications of Active Metabolites.
In: Journal of Medicinal Chemistry, 46
Artikel, Bibliographie

Schieffer, Bernhard ; Schmidt, Boris ; Drexler, H. (2003)
Angiotensin-II-Rezeptor-unabhängige anti-inflammatorische und antiaggregatorische Eigenschaften von AT1-Antagonisten. Rolle aktiver Metaboliten.
In: Herz BNK, 28
Artikel, Bibliographie

Schmidt, Boris (2003)
Aspartic Proteases involved in Alzheimer's disease.
In: ChemBioChem : a European journal of chemical biology, 4
Artikel, Bibliographie

Schmidt, Boris (2003)
Selective inhibition of proteases :design of beta- and gamma-scretase inhibitors.
Konferenzveröffentlichung, Bibliographie

Schmidt, Boris ; Kühn, Christian ; Ehlert, Dennis K. ; Lindeberg, Gunnar ; Lindman, Susanne ; Karlén, Anders ; Hallberg, Anders (2003)
A frame shifted disulfide bridged analogue of angiotensin II.
In: Bioorganic medicinal chemistry
Artikel, Bibliographie

2002

Krämer, Christine ; Sunkomat, Julia ; Witte, Jane ; Luchtefeld, Maren ; Walden, Michael ; Schmidt, Boris ; Boger, Rainer H. ; Tsikas, Dimitrios ; Forssmann, Wolf-Georg ; Drexler, Helmut ; Schieffer, Bernhard (2002)
Angiotensin II receptor-independent antiinflammatory and antiaggregatory properties of Losartan : role of the active metabolite EXP3179.
In: Circulation Research, 90
Artikel, Bibliographie