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Number of items: 32.

Stubba, Daniel and Bensinger, Dennis and Steinbacher, Janika and Proskurjakov, Lilia and Salcedo Gómez, Álvaro and Schmidt, Uwe and Roth, Stefan and Schmitz, Katja and Schmidt, Boris (2019):
Cell‐Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit.
In: ChemMedChem, (23), 14. pp. 2005-2022, ISSN 1860-7179,
DOI: 10.1002/cmdc.201900472,
[Online-Edition: https://doi.org/10.1002/cmdc.201900472],
[Article]

Bensinger, Dennis and Stubba, Daniel and Cremer, Anjali and Kohl, Vanessa and Waßmer, Theresa and Stuckert, Johanna and Engemann, Victoria and Stegmaier, Kimberly and Schmitz, Katja and Schmidt, Boris (2019):
Virtual Screening Identifies Irreversible FMS-like Tyrosine Kinase 3 Inhibitors with Activity toward Resistance-Conferring Mutations.
In: Journal of Medicinal Chemistry, (5), 62. American Chemical Society, pp. 2428-2446, ISSN 0022-2623,
DOI: 10.25534/tuprints-00009651,
[Online-Edition: https://tuprints.ulb.tu-darmstadt.de/9651],
[Article]

Bensinger, Dennis and Neumann, Theresa and Scholz, Christoph and Voss, Constantin and Knorr, Sabine and Kuckelkorn, Ulrike and Hamacher, Kay and Kloetzel, Peter-Michael and Schmidt, Boris (2016):
Elastase-like Activity Is Dominant to Chymotrypsin-like Activity in 20S Proteasome's β5 Catalytic Subunit.
In: ACS chemical biology, 11 (7), pp. 1800-1804, ISSN 1554-8937,
[Article]

Scholz, Christoph and Knorr, Sabine and Hamacher, Kay and Schmidt, Boris (2015):
DOCKTITE-A Highly Versatile Step-by-Step Workflow for Covalent Docking and Virtual Screening in the Molecular Operating Environment.
In: Journal of chemical information and modeling, 55 (2), pp. 398-406, ISSN 1549-960X,
[Article]

Neumann, Theresa and Benajiba, Lina and Göring, Stefan and Stegmaier, Kimberly and Schmidt, Boris (2015):
Evaluation of Improved Glycogen Synthase Kinase-3α Inhibitors in Models of Acute Myeloid Leukemia.
In: Journal of Medicinal Chemistry, (22), 58. American Chemical Society, pp. 8907-8919, ISSN 0022-2623,
DOI: 10.25534/tuprints-00009652,
[Online-Edition: https://tuprints.ulb.tu-darmstadt.de/9652],
[Article]

Voss, Constantin and Scholz, Christoph and Knorr, Sabine and Beck, Philipp and Stein, Martin L. and Zall, Andrea and Kuckelkorn, Ulrike and Kloetzel, Peter-Michael and Groll, Michael and Hamacher, Kay and Schmidt, Boris (2014):
α-Keto Phenylamides as P1'-Extended Proteasome Inhibitors.
In: ChemMedChem, 9 (11), pp. 2557-2564, ISSN 1860-7187,
[Article]

Schupp, M. and Lee, C. L. D. and Frost, N. and Umbreen, Sumaira and Schmidt, Boris and Unger, T. and Kintscher, U. (2006):
CHBPR-Regulation of PPARg Activity by Losartan Metabolites.
In: Hypertension, 47pp. 586-589, [Article]

Everson da Silva, Luiz and Joussef, Antonio Carlos and Foro, Sabine and Schmidt, Boris (2005):
4-Fluoro-N-(quinolin-8-yl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, (12), 61. Wiley, pp. o4387-o4388, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805039188,
[Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
4-Nitro-N-(8-quinolyl)-benzenesulfon-amide.
In: Acta Crystallographica, Section E: Structure Reports Online, (11), 61. Wiley, pp. o3778-o3779, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805032691,
[Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
5 2,4,6-Triisopropyl-N-(8-quinolyl)-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, (11), 61. Wiley, pp. o3780-o3781, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805032708,
[Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
N-(5,7-Dibromo-8-quinolyl)-4-fluoro-benzenesulfonamide.
In: Acta Crystallographica, Section E: Structure Reports Online, (11), 61. Wiley, pp. o3782-o3783, e-ISSN 1600-5368,
DOI: 10.1107/S160053680503271X,
[Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
5,7-Dibromo-N-tosyl-quinolin-8-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, (10), 61. Wiley, pp. o3435-o3436, e-ISSN 1600-5368,
DOI: 10.1107/S160053680502773X,
[Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
6-Nitroquinolin-2(1H)-one.
In: Acta Crystallographica, Section E: Structure Reports Online, (9), 61. Wiley, pp. o2992-o2993, e-ISSN 1600-5368,
DOI: 10.1107/S1600536805025894,
[Article]

Braun, Hannes R. and Meusinger, Reinhard and Schmidt, Boris (2005):
2-iodethanols from aldehydes, diiodomethane and iso-propylmagnesium chloride.
In: Tetrahedron Letters, 46pp. 2551-2554, [Article]

Schmidt, Boris and Narlawar, Rajeshwar and Braun, Hannes (2005):
Drug Development and PET-Diagnostics for Alzheimer's Disease.
In: Current Medicinal Chemistry, 12pp. 1677-1695, [Article]

Everson da Silva, Luiz and Joussef, Antonio C. and Foro, Sabine and Schmidt, Boris (2005):
N-Benzyl-8-nitroquinolin-2-amine.
In: Acta Crystallographica, Section E: Structure Reports Online, 61pp. o3837-o3838, [Article]

Braun, A. and Umbreen, Sumaira and Groll, M. and Kuckelkorn, U. and Mlynarczuk, I. and Wiegand, M. E. and Drung, I. and Kloetzel, P. M. and Schmidt, Boris (2005):
Tripeptide mimetics inhibit the 20S proteasome by covalent bonding to the active site threonines.
In: Journal of Biological Chemistry, 280pp. 28394-28411, [Article]

Schmidt, Boris and Siegler, Alexander (2004):
Aspartic Proteases involved in Alzheimer's disease.
In: Highlights in bioorganic chemistry. Eds.: Schmuck, Carsten ; Wennemers, Helma. - Weinheim : Wiley-VCH Verl. , 2004. S. 262-276 , ISBN 3-527-30656-0, Weinheim, Wiley-VCH Verl., [Book Section]

Schmidt, Boris and Jiricek, Jan and Titz, Alexander and Ye, Guofeng and Parang, Keykavous (2004):
Copper dipicolinates as peptidomimetic ligands for the Src SH2 domain.
In: Bioorganic & Medicinal Chemistry Letters, 14pp. 4203-4206, [Article]

Schmidt, Boris and Braun, Hannes A. (2004):
E-1,2-Dichlorovinyl ethers as irreversible protease inhibitors.
In: Tetrahydron Letterrs, 45pp. 1751-1753, [Article]

Larbig, Gregor and Zall, Andreas and Schmidt, Boris (2004):
Inhibitors designed for presenilin 1 by means of aspartic acid activation : Preliminary Communication.
In: Helvetica Chimica Acta, 87pp. 2334-2340, [Article]

Schmidt, Boris (2004):
[Rez.:] Molecular biology in medicinal chemistry / ed. by Th. Dingermann .... - Weinheim : Wiley-VCH, 2004 (Methods and principles in medicinal chemistry ; 21) ISBN 7-30431-2.
In: ChemBioChem, 5pp. 1153-1154, [Article]

Schmidt, Boris and Larbig, Gregor (2004):
[Rez.:] More targets, strategies, methods / K. C. Nicolaou and S. A. Snyder. - 2003. -(Classics in total synthesis / K. C. Nicolaou and S. A. Snyder ; 2) ISBN: 3-527-30685-4.
In: ChemBioChem (ISSN 1439-4227), 5p. 885, [Article]

Schmidt, Boris and Drexler, H. and Schieffer, Bernhard (2004):
Therapeutic Effects of Angiotensin (AT1) Receptor Antagonists: Potential Contribution of Mechanisms Other Than AT1 Receptor Blockade.
In: American Journal of Cardiovascular Drugs, pp. 361-368, [Article]

Schmidt, Boris and Drexler, Helmut and Schieffer, Bernhard (2004):
Therapeutic effects of angiotensin (AT1) receptor antagonists : potential contribution of mechanisms other than AT1 receptor blockade.
In: American Journal of Cardiovascular Drugs, 4pp. 361-368, [Article]

Muller, Gilles and Schmidt, Boris and Jiricek, Jan and Lbuenzli, Jean Claude G. and Schenk, Kurt J. (2003):
3-[2,6-Bis(diethyl-carbamoyl)-pyridin-4-yl]-N-(tert-butoxycarbonyl)alanine methyl ester: a chiral tridentate ligand that causes a diastereomeric excess of its lanthanide complexes in solution.
In: Acta Crystallographica, Section C: Crystal Structure Communications, 59pp. 353-356, [Article]

Schmidt, Boris and Schieffer, Bernhard (2003):
Angiotensin II AT1 Receptor Antagonists : Clinical Implications of Active Metabolites.
In: Journal of Medicinal Chemistry, 46p. 2261, [Article]

Schieffer, Bernhard and Schmidt, Boris and Drexler, H. (2003):
Angiotensin-II-Rezeptor-unabhängige anti-inflammatorische und antiaggregatorische Eigenschaften von AT1-Antagonisten. Rolle aktiver Metaboliten.
In: Herz BNK, 28p. 2, [Article]

Schmidt, Boris (2003):
Aspartic Proteases involved in Alzheimer's disease.
In: ChemBioChem : a European journal of chemical biology, 4pp. 367-378, [Article]

Schmidt, Boris (2003):
Selective inhibition of proteases :design of beta- and gamma-scretase inhibitors.
In: International conference on aspartic proteases and inhibitors <2003, Kyoto, Japan> : [proceedings], S. 20, [Conference or Workshop Item]

Schmidt, Boris and Kühn, Christian and Ehlert, Dennis K. and Lindeberg, Gunnar and Lindman, Susanne and Karlén, Anders and Hallberg, Anders (2003):
A frame shifted disulfide bridged analogue of angiotensin II.
In: Bioorganic medicinal chemistry, pp. 985-990, [Article]

Krämer, Christine and Sunkomat, Julia and Witte, Jane and Luchtefeld, Maren and Walden, Michael and Schmidt, Boris and Boger, Rainer H. and Tsikas, Dimitrios and Forssmann, Wolf-Georg and Drexler, Helmut and Schieffer, Bernhard (2002):
Angiotensin II receptor-independent antiinflammatory and antiaggregatory properties of Losartan : role of the active metabolite EXP3179.
In: Circulation Research, 90. pp. 770-777, [Article]

This list was generated on Tue Jun 2 02:21:09 2020 CEST.